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Ngwaahịa

Doramectin 117704-25-3 Ọgwụ mgbochi ọrịa parasitic

Nkọwa dị mkpirikpi:

Ụdị okwu:25-Cclohexyl-avermectin B1, Avermectin A1a

Nọmba CAS:117704-25-3

Ogo:n'ụlọ

Ụdị molekụla:C50H74O14

Ibu Formula:899.11


Nkọwa ngwaahịa

Mkpado ngwaahịa

Ụgwọ:T/T, L/C
Isi mmalite ngwaahịa:China
Ọdụ ụgbọ mmiri:Beijing/Shanghai/Hangzhou
Ike mmepụta:15kg / ọnwa
Nye iwu (MOQ):1 n'arọ
Etiti oge:3 ụbọchị ọrụ
Ọnọdụ nchekwa:Chekwaa na okpomọkụ 2-8 ℃ maka ogologo oge, na-echebe site na ìhè.
Ihe ngwugwu:karama
Nha ngwugwu:1kg/drum
Ozi nchekwa:UN 2811 6.1 / PG 3

Doramectin

Okwu mmalite

Dorametin bụ ọgwụ antiparasitic ọgbọ ọhụrụ macrolide.Ọ bụ ọgwụ nje avermectin na-emepụta site na gbaa ụka nke ụdị ọhụrụ Streptomyces avermitis na cyclohexamic acid dị ka ihe mbụ.A na-ewere ya dị ka otu n'ime ọgwụ antiparasitic kacha mma na ezinụlọ avermectin.

Mmetụta ụmụ ahụhụ nke Doramectin yiri Ivermectin, nke nwere ike igbochi nnyefe nke mkpali akwara n'etiti akwara na mọzụlụ, ma mee ka ahụhụ ahụ kpọnwụrụ akpọnwụ wee nwụọ n'ebe onye ọbịa ahụ nọ.Otú ọ dị, n'ihi ụbara ọbara dị elu nke doramectin n'ime ahụ, mkpochapụ ahụ na-adị nwayọọ nwayọọ, na oge nlekọta nke ịdị irè na-adịte aka, ya mere mmetụta nke ụmụ ahụhụ dị mma karịa Ivermectin.N'ihi enweghị mmeghachi ahụ nfụkasị ahụ mgbe ị na-eji Doramectin, ya mere ọ dị nchebe karịa ka a ga-eji.A na-ewerekwa ya dị ka ọgwụ nke kama Ivermectin.

A na-eji ya maka ọgwụgwọ na ịchịkwa parasitosis dị n'ime (gastrointestinal nematodes na pulmonary nematodes), akọrọ na mange (na ndị ọzọ ectoparasites).

Clinically na-egosi na Doramectin nwere mmetụta dị mma na nematodes na tract digestive nke ezì.Dị ka akụkọ ahụ si kwuo, a na-enye ezì intramuscularly na dose nke 0.3 mg / kg arọ ahụ.Ọnụ ọgụgụ dị arọ nke ọrịa artificial na ọrịa ọrịa anụ ahụ dị elu karịa nke ndị na-achịkwa na 7, 14 na 21 ụbọchị mgbe nchịkwa gasịrị.N'iji ya tụnyere otu njikwa, a na-ewepụ ikpuru 100% na-enweghị mmetụta ọ bụla.

Ọ na-egosikwa ụlọ ọgwụ na ọgwụgwọ Sarcoptes scabies, enwere mmetụta dị mma site na piglets na-aṅụ ara na-akụ.

Doramectin dịkwa maka ịnyịnya dị ka ọnụ, ekpomeekpo, gel bioadhesive n'okpuru aha.

Doramectin anaghị eguzosi ike na okike.Ọ na-emebi ngwa ngwa ma ghara ime ya n'okpuru ìhè anyanwụ.Ọgwụ ndị fọdụrụnụ na-egbu egbu nye azụ̀ na ihe ndị dị n'ime mmiri.Ya mere, ekwesịrị ịṅa ntị na nchebe mmiri.

Nkọwapụta (N'ụlọ Ọkọlọtọ)

Ihe

Nkọwapụta

Ọdịdị White crystalline ntụ ntụ
njirimara HPLC, IR
Ọdịdị nke ngwọta Ihe ngwọta doro anya na ọ bụghị ihe siri ike na agba karịa ntụaka ngwọta BY6
Mmiri ≤3%
Igwe dị arọ ≤20ppm
Sulfated Ash ≤0.1%
BHT ≤2000ppm
Ihe metụtara ya Avermectin B1a ≤1.5%
Avermectin B1b≤1.0%
Avermectin B1a na Avermectin B1b≤2.0%
Mkpokọta adịghị ọcha NMT 5.0%
Ihe mgbaze fọdụrụnụ acetone ≤5000ppm
Ethanol≤30000ppm
Ethyl acetate ≤5000ppm
Methanol≤3000ppm
Nyocha ≥95% (na anhydrous na ihe mgbaze free ndabere)

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