The Laboratory tubes

Ngwaahịa

Posaconazole 171228-49-2 ọgwụ nje

Nkọwa dị mkpirikpi:

Ụdị okwu:Noxafil;56592

Nọmba CAS:171228-49-2

Ogo:n'ụlọ

Ụdị molekụla:C43H66N12O12S2

Ibu Formula:700.78


Nkọwa ngwaahịa

Mkpado ngwaahịa

Ụgwọ:T/T, L/C
Isi mmalite ngwaahịa:China
Ọdụ ụgbọ mmiri:Beijing/Shanghai/Hangzhou
Ike mmepụta:20kg / ọnwa
Nye iwu (MOQ):10g
Etiti oge:3 ụbọchị ọrụ
Ọnọdụ nchekwa:Echekwara ya na ebe dị jụụ, ebe akọrọ, okpomọkụ ụlọ.
Ihe ngwugwu:vial
Nha ngwugwu:10g / vial
Ozi nchekwa:Ọ bụghị ngwongwo dị ize ndụ

Posaconazole

Okwu mmalite

Posaconazole bụ ọgwụ antifungal nke triazole.
A na-eji Posaconazole agwọ ọrịa Aspergillus na Candida.A na-ejikwa ya maka ọgwụgwọ nke oropharyngeal candidiasis (OPC), gụnyere OPC refractory to itraconzaole na/ma ọ bụ ọgwụgwọ fluconazole.
A na-ejikwa ya na-agwọ ọrịa na-efe efe site na Candida, Mucor, na Aspergillus ụdị n'ime ndị ọrịa nwere nnukwu mgbochi.

Nkọwapụta (ọkọlọtọ n'ụlọ)

Ihe

Nkọwapụta

Ọdịdị White ma ọ bụ ihe fọrọ nke nta ka ọ bụrụ ọcha, hygroscopic ntụ ntụ

Ihe

Nkọwapụta

Ọdịdị

Uzuzu crystalline ọcha ma ọ bụ na-acha ọcha

Ntughari pụrụ iche

-28.0°~-34.0°

Ụdị kristal

Ọ kwesịrị ịbụ kristal Ⅰ, nwere akụkụ 2-theta nke

14.4±0.2°,19.2±0.2°,21.7±0.2°,24.3±0.2°29.3±0.2°

njirimara

IR, HPLC

Ihe ndị emetụtara I

PO-R1 NMT 0.10%

PO-R2 NMT 0.10%

PO-R3 NMT 0.10%

PO-R4 NMT 0.10%

PO-D3 & PO-D5 NMT 0.10%

PO-D7 & PO-D10 NMT 0.10%

Nke ọ bụla n'ime adịghị ọcha NMT 0.10%

Mkpokọta adịghị ọcha NMT 0.5%

Ihe ndị metụtara Ⅱ

PO-E NMT 0.10%

PO-D1 NMT 0.10%

PO-R5 NMT 0.10%

Ihe mgbaze fọdụrụnụ

Methanol NMT 3000ppm

Ethanol NMT 5000ppm

Dichloromethane NMT 600ppm

Tetrahydrofuran NMT 720ppm

N, N-dimethyl formamide NMT 880ppm

Triethylamine NMT 100ppm

Dimethy sulfoxide NMT 5000ppm

Mmiri

NMT 2.0%

Ihe fọdụrụ na mgbanye

NMT 0.1%

Ọla dị arọ

NMT 10pm

Oke microbial

Mkpokọta ikuku ikuku NMT 1000cfu/g

Mkpokọta yist na ebu NMT 100cfu/g

E.coli kwesịrị ịpụ

Nyocha

98.0% -102.0% (na-esighi ike)

98.0% -102.0% (na anhydrous na ihe mgbaze n'efu)


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