The Laboratory tubes

Ngwaahịa

Pimobendan 74150-27-9 Metabolism PDE inhibitor

Nkọwa dị mkpirikpi:

Aha ngwaahịa:Pimobendan
Ụdị okwu:4,5-Dihydro-6-[2- (4-methoxyphenyl) -1H-benzimizol-6-yl] -5-methyl-3 (2H) -pyridazinone.
Nọmba CAS:74150-27-9
Ogo:USP43
Usoro ihe omimi:C19H18N4O2
Arọ molikula:334.37


Nkọwa ngwaahịa

Mkpado ngwaahịa

Ụgwọ:T/T, L/C
Isi mmalite ngwaahịa:China
Ọdụ ụgbọ mmiri:Beijing/Shanghai/Hangzhou
Nye iwu (MOQ):1g
Etiti oge:3 ụbọchị ọrụ
Ike mmepụta:1kg / ọnwa
Ọnọdụ nchekwa:Echekwara ya na ebe dị jụụ, ebe akọrọ, okpomọkụ ụlọ.
Ihe ngwugwu:vial, karama
Nha ngwugwu:1g / vial, 5/vial, 10g / vial, 50g / karama, 500g / karama
Ozi nchekwa:UN 2811 6.1/PG 3

Pimobendan

Okwu mmalite

Pimobendan, bụ ọgwụ anụmanụ.Ọ bụ ihe mmetụta calcium na onye na-emechi phosphodiesterase 3 (PDE3) nwere mmetụta inotropic na vasodilator dị mma.

A na-eji Pimobendan na njikwa nkụda obi na nkịta, nke na-ebutekarị ọrịa myxomatous mitral valve (nke a na-akpọbu endocardiosis), ma ọ bụ cardiomyopathy dilated.Nnyocha egosila na dị ka monotherapy, pimobendan na-abawanye oge ịlanarị ma na-eme ka ndụ dịkwuo mma na ndị ọrịa canine nwere nkụchi obi nke abụọ na ọrịa mitral valvụ ma e jiri ya tụnyere benazepril, onye na-egbochi ACE.

Nkọwapụta (USP43)

Ihe

Nkọwapụta

Ọdịdị

White ma ọ bụ ubé odo ntụ ntụ, hygroscopic

Mp

Ihe dịka 242 ℃

Solubility

Ihe na-adịghị ahụkebe n'ime mmiri, na-agbaze kpamkpam na dimethylformamide, soluble ntakịrị na acetone yana na methanil.

njirimara

Infrared absorption spectrophotometry, atụnyere pimobendan CRS.

Oge njide nke isi kacha elu nke ngwọta Sample dabara na nke Standard ngwaahịa ngwọta, dị ka enwetara na Organic adịghị ọcha ule.

Ọla dị arọ

≤10ppm

Ọkpụkpụ granularity

P90 ≤ 25μm

Nha urughuru

20-80 ntupu

Ihe mgbaze fọdụrụnụ

≤500ppm

Mmiri

≤ 1.0%

Nyocha

98.0% ~ 102.0%

Sulfated uyi

≤0.10%

Ihe ndị emetụtara (HPLC)

adịghị ọcha A

≤0.10%

adịghị ọcha B

≤0.10%

Ọdịghị ọcha ọ bụla ọzọ

≤0.10%

Mkpokọta adịghị ọcha

≤0.20%


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